6beta-[N,N-Bis(2-chloroethyl)amino]-17-(cyclopropylmethyl)-4,5alpha-epoxy-3,14-dihydroxymorphinan(chlornaltrexamine) a potent opioid receptor alkylating agent with ultralong narcotic antagonist actitivty.
D000477:Alkylating Agents / Q000138:chemical synthesis* / Q000494:pharmacology; D000698:Analgesia; D001667:Binding, Competitive; D009020:Morphine / Q000037:antagonists & inhibitors; D009270:Naloxone / Q000031:analogs & derivatives*; D009271:Naltrexone / Q000031:analogs & derivatives* / Q000138:chemical synthesis / Q000494:pharmacology; D009292:Narcotic Antagonists / Q000138:chemical synthesis*; D009588:Nitrogen Mustard Compounds / Q000138:chemical synthesis / Q000494:pharmacology; D011957:Receptors, Opioid / Q000187:drug effects*
D000477:Alkylating Agents; D009292:Narcotic Antagonists; D009588:Nitrogen Mustard Compounds; D011957:Receptors, Opioid; D009270:Naloxone; D009271:Naltrexone; C017120:chlornaltrexamine; D009020:Morphine