In vitro evaluation of a casomorphin related pentapeptide, a competitive mu opioid receptor antagonist.
Davis
P
P
Department of Pharmacology, University of Arizona, Tucson 85724.
Tourwe
D
D
Delaet
N
N
Kramer
T H
TH
Burks
T F
TF
D000595:Amino Acid Sequence; D000818:Animals; D001667:Binding, Competitive / Q000187:drug effects; D004723:Endorphins / Q000037:antagonists & inhibitors / Q000138:chemical synthesis / Q000494:pharmacology*; D020881:Enkephalin, D-Penicillamine (2,5)-; D004745:Enkephalins / Q000494:pharmacology; D006168:Guinea Pigs; D007082:Ileum / Q000187:drug effects; D066298:In Vitro Techniques; D008297:Male; D051379:Mice; D008813:Mice, Inbred ICR; D008969:Molecular Sequence Data; D009119:Muscle Contraction / Q000187:drug effects; D009130:Muscle, Smooth / Q000187:drug effects; D009292:Narcotic Antagonists; D017450:Receptors, Opioid, mu; D014649:Vas Deferens / Q000187:drug effects
D004723:Endorphins; D004745:Enkephalins; D009292:Narcotic Antagonists; D017450:Receptors, Opioid, mu; C072948:CM 2-3; C021968:beta-casomorphins; C044708:morphiceptin, N-Me-Phe(3)-; D020881:Enkephalin, D-Penicillamine (2,5)-