title: Peptides incorporating electrophilic glutamine analogues as potential transglutaminase inhibitors.
authors.affiliation: Department of Medicinal Chemistry, Wellcome Research Laboratories, Beckenham, Kent, U.K.
authors.forename: P M
authors.initials: PM
authors.lastname: Doyle
authors.forename: C J
authors.initials: CJ
authors.lastname: Harris
authors.forename: K R
authors.initials: KR
authors.lastname: Carter
authors.forename: D S
authors.initials: DS
authors.lastname: Simpkin
authors.forename: P
authors.initials: P
authors.lastname: Bailey-Smith
authors.forename: D
authors.initials: D
authors.lastname: Stone
authors.forename: L
authors.initials: L
authors.lastname: Russell
authors.forename: G J
authors.initials: GJ
authors.lastname: Blackwell
mesh_terms: D000595:Amino Acid Sequence; D005973:Glutamine / Q000031:analogs & derivatives; D006801:Humans; D066298:In Vitro Techniques; D007700:Kinetics; D008969:Molecular Sequence Data; D010455:Peptides / Q000737:chemistry / Q000378:metabolism / Q000494:pharmacology*; D013329:Structure-Activity Relationship; D013379:Substrate Specificity; D011503:Transglutaminases / Q000037:antagonists & inhibitors* / Q000378:metabolism
chemical_list: D010455:Peptides; D005973:Glutamine; D011503:Transglutaminases