Novel photoaffinity label for the dopamine D2 receptor: synthesis of 4-azido-5-iodo-2-methoxy-N-[1-(phenylmethyl)-4-piperidinyl] benzamide (iodoazidoclebopride, IAC) and the corresponding 125I-labeled analogue (125IAC).
Neumeyer
J L
JL
Guan
J H
JH
Niznik
H B
HB
Dumbrille-Ross
A
A
Seeman
P
P
Padmanabhan
S
S
Elmaleh
D R
DR
D000345:Affinity Labels / Q000138:chemical synthesis* / Q000378:metabolism; D000818:Animals; D001386:Azides / Q000138:chemical synthesis* / Q000378:metabolism; D001549:Benzamides / Q000138:chemical synthesis* / Q000378:metabolism; D007457:Iodine Radioisotopes; D010782:Photolysis; D051381:Rats; D011954:Receptors, Dopamine / Q000378:metabolism*; D017448:Receptors, Dopamine D2
D000345:Affinity Labels; D001386:Azides; D001549:Benzamides; D007457:Iodine Radioisotopes; D011954:Receptors, Dopamine; D017448:Receptors, Dopamine D2; C044896:4-azido-5-iodoclebopride