Structure-activity relationships in 1,2,3-triazol-1-yl derivatives of clavulanic acid.
The synthesis of a series of analogues of clavulanic acid, possessing a substituted 1,2,3-triazole ring in place of the exocyclic hydroxyl group, is described. Quantitative structure-activity relationships in this series are discussed.
D002969:Clavulanic Acids / Q000494:pharmacology*; D009682:Magnetic Resonance Spectroscopy; D008826:Microbial Sensitivity Tests; D013329:Structure-Activity Relationship
D002969:Clavulanic Acids