Variations in affinities for the NK1 receptor: differences between the non-peptide substance P antagonists RP 67580 and CP-96,345 and the agonist septide.
Fardin
V
V
Biology Department, Rhone-Poulenc Rorer, Centre de Recherches de Vitry-Alfortville, Vitry sur Seine, France.
Foucault
F
F
Bock
M D
MD
Jolly
A
A
Flamand
O
O
Clerc
F
F
Garret
C
C
D000818:Animals; D001667:Binding, Competitive; D001713:Biphenyl Compounds / Q000378:metabolism*; D001921:Brain / Q000378:metabolism*; D002460:Cell Line; D004285:Dogs; D006168:Guinea Pigs; D006801:Humans; D007211:Indoles / Q000378:metabolism*; D054833:Isoindoles; D051379:Mice; D010446:Peptide Fragments / Q000378:metabolism*; D011761:Pyrrolidonecarboxylic Acid / Q000031:analogs & derivatives; D051381:Rats; D018040:Receptors, Neurokinin-1 / Q000378:metabolism*; D013363:Submandibular Gland / Q000378:metabolism; D013373:Substance P / Q000031:analogs & derivatives* / Q000037:antagonists & inhibitors* / Q000378:metabolism*
D001713:Biphenyl Compounds; D007211:Indoles; D054833:Isoindoles; D010446:Peptide Fragments; D018040:Receptors, Neurokinin-1; C071693:7,7-diphenyl-2-(1-imino-2-(2-methoxyphenyl)ethyl)perhydroisoindol-4-one; D013373:Substance P; C054725:septide; D011761:Pyrrolidonecarboxylic Acid; C066892:CP 96345