title: 2-Phenyl-4-quinolinecarboxamides: a novel class of potent and selective non-peptide competitive antagonists for the human neurokinin-3 receptor.
authors.affiliation: Department of Chemistry, SmithKline Beecham S.p.A., Milano, Italy.
authors.forename: G A
authors.initials: GA
authors.lastname: Giardina
authors.forename: H M
authors.initials: HM
authors.lastname: Sarau
authors.forename: C
authors.initials: C
authors.lastname: Farina
authors.forename: A D
authors.initials: AD
authors.lastname: Medhurst
authors.forename: M
authors.initials: M
authors.lastname: Grugni
authors.forename: J J
authors.initials: JJ
authors.lastname: Foley
authors.forename: L F
authors.initials: LF
authors.lastname: Raveglia
authors.forename: D B
authors.initials: DB
authors.lastname: Schmidt
authors.forename: R
authors.initials: R
authors.lastname: Rigolio
authors.forename: M
authors.initials: M
authors.lastname: Vassallo
authors.forename: V
authors.initials: V
authors.lastname: Vecchietti
authors.forename: D W
authors.initials: DW
authors.lastname: Hay
mesh_terms: D000818:Animals; D001667:Binding, Competitive; D016466:CHO Cells; D002924:Ciliary Body / Q000187:drug effects; D006224:Cricetinae; D003412:Cricetulus; D015195:Drug Design; D006168:Guinea Pigs; D006801:Humans; D009119:Muscle Contraction / Q000187:drug effects; D010446:Peptide Fragments / Q000037:antagonists & inhibitors; D010880:Piperidines / Q000737:chemistry / Q000494:pharmacology; D011804:Quinolines / Q000737:chemistry / Q000145:classification / Q000494:pharmacology*; D011817:Rabbits; D018042:Receptors, Neurokinin-3 / Q000037:antagonists & inhibitors*; D011993:Recombinant Fusion Proteins / Q000037:antagonists & inhibitors; D013329:Structure-Activity Relationship; D013373:Substance P / Q000031:analogs & derivatives / Q000037:antagonists & inhibitors
chemical_list: D010446:Peptide Fragments; D010880:Piperidines; D011804:Quinolines; D018042:Receptors, Neurokinin-3; D011993:Recombinant Fusion Proteins; C054724:senktide; D013373:Substance P; C091554:SR 142801