New bradykinin antagonists having very high potency at B1 receptors.
Gera
L
L
Department of Biochemistry University of Colorado School of Medicine, Denver 80262, USA.
Stewart
J M
JM
Whalley
E T
ET
Burkard
M
M
Zuzack
J S
JS
D000595:Amino Acid Sequence; D000818:Animals; D001011:Aorta / Q000187:drug effects / Q000502:physiology; D001920:Bradykinin / Q000037:antagonists & inhibitors* / Q000737:chemistry / Q000378:metabolism; D016466:CHO Cells; D002460:Cell Line; D006224:Cricetinae; D006168:Guinea Pigs; D006801:Humans; D007082:Ileum / Q000378:metabolism; D066298:In Vitro Techniques; D015394:Molecular Structure; D009842:Oligopeptides / Q000737:chemistry / Q000378:metabolism* / Q000494:pharmacology*; D011817:Rabbits; D043783:Receptor, Bradykinin B1; D018002:Receptors, Bradykinin / Q000378:metabolism*; D013329:Structure-Activity Relationship; D014664:Vasodilation / Q000187:drug effects
D009842:Oligopeptides; D043783:Receptor, Bradykinin B1; D018002:Receptors, Bradykinin; D001920:Bradykinin