From histamine H2 receptor regulation to reclassification of H2 antagonists; inverse agonism as the basis for H2 receptor upregulation.
Smit
M J
MJ
Leiden/Amsterdam Center for Drug Research, Department of Pharmacochemistry, Vrije Universiteit, Amsterdam, The Netherlands.
Timmerman
H
H
Alewijnse
A E
AE
Leurs
R
R
D000818:Animals; D016466:CHO Cells; D002927:Cimetidine / Q000494:pharmacology*; D006224:Cricetinae; D006635:Histamine H2 Antagonists / Q000494:pharmacology*; D051381:Rats; D011970:Receptors, Histamine H2 / Q000235:genetics / Q000378:metabolism*
D006635:Histamine H2 Antagonists; D011970:Receptors, Histamine H2; D002927:Cimetidine