Reporter affinity labels: an o-phthalaldehyde derivative of beta-naltrexamine as a fluorogenic ligand for opioid receptors.
Le Bourdonnec
B
B
Department of Medicinal Chemistry, College of Pharmacy, School of Medicine, University of Minnesota, Minneapolis 55455, USA.
El Kouhen
R
R
Lunzer
M M
MM
Law
P Y
PY
Loh
H H
HH
Portoghese
P S
PS
D000345:Affinity Labels; D000818:Animals; D016466:CHO Cells; D006224:Cricetinae; D008024:Ligands; D051379:Mice; D009271:Naltrexone / Q000031:analogs & derivatives* / Q000138:chemical synthesis / Q000737:chemistry / Q000378:metabolism / Q000494:pharmacology; D009292:Narcotic Antagonists / Q000138:chemical synthesis* / Q000737:chemistry / Q000378:metabolism / Q000494:pharmacology; D010147:Pain Measurement; D011957:Receptors, Opioid / Q000378:metabolism*; D017465:Receptors, Opioid, delta / Q000378:metabolism; D017473:Receptors, Opioid, kappa / Q000378:metabolism; D017450:Receptors, Opioid, mu / Q000378:metabolism; D009764:o-Phthalaldehyde / Q000031:analogs & derivatives* / Q000138:chemical synthesis* / Q000737:chemistry / Q000378:metabolism
D000345:Affinity Labels; D008024:Ligands; D009292:Narcotic Antagonists; D011957:Receptors, Opioid; D017465:Receptors, Opioid, delta; D017473:Receptors, Opioid, kappa; D017450:Receptors, Opioid, mu; D009271:Naltrexone; D009764:o-Phthalaldehyde; C024524:beta-funaltrexamine