title: Synthesis and systemic fungicidal activity of silicon-containing azole derivatives.
abstract: A new series of azole derivatives containing silicon were synthesized and evaluated for fungicidal activity against rice sheath blight by submerged application. Among them, 2-(4-fluorophenyl)-1-(1H-1,2,4-triazol-1-yl)-3-trimethylsilylpr opan-2-ol (9a) exhibited satisfactory efficacy at 12.5 grams per 10 ares.
authors.affiliation: Agroscience Research Laboratories, Sankyo Co., Ltd., Siga, Japan. hiroit@yasu.sankyo.co.jp
authors.forename: H
authors.initials: H
authors.lastname: Itoh
authors.forename: R
authors.initials: R
authors.lastname: Yoneda
authors.forename: J
authors.initials: J
authors.lastname: Tobitsuka
authors.forename: T
authors.initials: T
authors.lastname: Matsuhisa
authors.forename: H
authors.initials: H
authors.lastname: Kajino
authors.forename: H
authors.initials: H
authors.lastname: Ohta
authors.forename: N
authors.initials: N
authors.lastname: Hayashi
authors.forename: Y
authors.initials: Y
authors.lastname: Takahi
authors.forename: M
authors.initials: M
authors.lastname: Tsuda
authors.forename: H
authors.initials: H
authors.lastname: Takeshiba
mesh_terms: D000935:Antifungal Agents / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D001393:Azoles / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D008826:Microbial Sensitivity Tests; D015394:Molecular Structure; D012275:Oryza / Q000382:microbiology; D012232:Rhizoctonia / Q000187:drug effects; D012825:Silicon / Q000737:chemistry*
chemical_list: D000935:Antifungal Agents; D001393:Azoles; D012825:Silicon