title: Phosphate-substituted ATP analogs are antagonists at human P2Y1 purinoceptors.
authors.affiliation: Institute of Chemical Physics, Tartu University, Estonia.
authors.forename: K
authors.initials: K
authors.lastname: Sak
authors.forename: G
authors.initials: G
authors.lastname: Raidaru
authors.forename: T E
authors.initials: TE
authors.lastname: Webb
authors.forename: J
authors.initials: J
authors.lastname: Järv
mesh_terms: D000244:Adenosine Diphosphate / Q000031:analogs & derivatives / Q000494:pharmacology; D000255:Adenosine Triphosphate / Q000031:analogs & derivatives* / Q000494:pharmacology; D000266:Adenylyl Imidodiphosphate / Q000494:pharmacology; D002460:Cell Line; D006801:Humans; D066298:In Vitro Techniques; D007295:Inositol Phosphates / Q000378:metabolism; D007700:Kinetics; D058919:Purinergic P2 Receptor Antagonists; D058472:Receptors, Purinergic P2Y1; D013873:Thionucleotides / Q000494:pharmacology
chemical_list: D007295:Inositol Phosphates; C546382:P2RY1 protein, human; D058919:Purinergic P2 Receptor Antagonists; D058472:Receptors, Purinergic P2Y1; D013873:Thionucleotides; D000266:Adenylyl Imidodiphosphate; C005147:5'-adenylyl (beta,gamma-methylene)diphosphonate; C002480:methylthio-ADP; D000244:Adenosine Diphosphate; D000255:Adenosine Triphosphate; C002630:alpha,beta-methyleneadenosine 5'-triphosphate