title: Covalently induced activation of the delta opioid receptor by a fluorogenic affinity label, 7'-(phthalaldehydecarboxamido)naltrindole (PNTI).
authors: Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota 55455, USA.
authors: B
authors: B
authors: Le Bourdonnec
authors: R
authors: R
authors: El Kouhen
authors: G
authors: G
authors: Poda
authors: P Y
authors: PY
authors: Law
authors: H H
authors: HH
authors: Loh
authors: D M
authors: DM
authors: Ferguson
authors: P S
authors: PS
authors: Portoghese
mesh_terms: D000345:Affinity Labels / Q000138:chemical synthesis* / Q000378:metabolism / Q000494:pharmacology; D000700:Analgesics / Q000138:chemical synthesis / Q000378:metabolism / Q000494:pharmacology; D000818:Animals; D016466:CHO Cells; D006224:Cricetinae; D005456:Fluorescent Dyes / Q000138:chemical synthesis* / Q000378:metabolism / Q000494:pharmacology; D006168:Guinea Pigs; D007082:Ileum / Q000187:drug effects / Q000502:physiology; D066298:In Vitro Techniques; D008024:Ligands; D008297:Male; D051379:Mice; D008958:Models, Molecular; D009271:Naltrexone / Q000031:analogs & derivatives / Q000138:chemical synthesis* / Q000378:metabolism / Q000494:pharmacology; D017465:Receptors, Opioid, delta / Q000819:agonists* / Q000378:metabolism; D014649:Vas Deferens / Q000187:drug effects / Q000502:physiology
chemical_list: C424722:17-(cyclopropylmethyl)-4,5-epoxy-3,4-dihydroxy-6-((phthalaldehydecarboxamido)acetamido)morphinan; D000345:Affinity Labels; D000700:Analgesics; D005456:Fluorescent Dyes; D008024:Ligands; D017465:Receptors, Opioid, delta; D009271:Naltrexone