Simple and convenient preparation of 1-(arylamino)methylbenzotriazoles and -(arylamino)methylbenzimidazoles.
The preparation of 1-(arylamino)methylbenzotriazoles 1a-17a and benzimidazoles 1b-17b is described and their antibacterial activity evaluated. 1-Hydroxymethylbenzazo-les react with the appropriate aniline to yield the target compounds. These were characterized using 1H NMR, IR, UV spectra. The compounds displayed no significant antibacterial activity.
Milata
V
V
Department of Organic Chemistry, Central Laboratory of Chemical Technique, Faculty of Chemical Technology, Slovak Republic.
Kada
R
R
Zalibera
L
L
Belicová
A
A
D001407:Bacillus / Q000378:metabolism; D001562:Benzimidazoles / Q000138:chemical synthesis*; D013055:Spectrophotometry, Infrared; D013056:Spectrophotometry, Ultraviolet; D014230:Triazoles / Q000138:chemical synthesis*
D001562:Benzimidazoles; D014230:Triazoles