title: Designing non-peptide peptidomimetics in the 21st century: inhibitors targeting conformational ensembles.
authors.affiliation: Department of Chemistry, University of Wisconsin-Madison, Madison, Wisconsin 53706, USA.
authors.forename: Matthew G
authors.initials: MG
authors.lastname: Bursavich
authors.forename: Daniel H
authors.initials: DH
authors.lastname: Rich
mesh_terms: D016282:Aspartic Acid Endopeptidases / Q000737:chemistry; D001665:Binding Sites; D015195:Drug Design; D004791:Enzyme Inhibitors / Q000737:chemistry*; D008024:Ligands; D008958:Models, Molecular; D018716:Molecular Mimicry; D010455:Peptides / Q000737:chemistry*; D011480:Protease Inhibitors / Q000737:chemistry; D011485:Protein Binding; D011487:Protein Conformation; D013329:Structure-Activity Relationship
chemical_list: D004791:Enzyme Inhibitors; D008024:Ligands; D010455:Peptides; D011480:Protease Inhibitors; D016282:Aspartic Acid Endopeptidases