Diastereoselective cascade synthesis of azabicyclo[3.1.0]hexanes from acyclic precursors.
The diastereoselective synthesis of azabicyclo[3.1.0]hexanes bearing different substituents on all positions of the cyclopropane ring has been achieved in moderate to good yields.
Molecular Innovation, Diversity and Automated Synthesis (MIDAS) Centre, School of Chemistry, Leeds University, Leeds, UK LS2 9JT.
Jutta
J
Böhmer
Ronald
R
Grigg
John D
JD
Marchbank