Synthesis of new alpha-heterocyclic alpha-aminoesters.
alpha-Heterocyclic alpha-aminoesters were obtained in good yields by reaction of a glycine cation equivalent and different heterocyclic nucleophiles; diastereoselectivity using a carbohydrate (galactopyranose) as N-protecting group was modest.
Bentama
A
A
Laboratoire de Chimie Organique, Faculté des Sciences et Techniques Fès-Saïss, Fès Maroc.
El Hadrami
E M
EM
El Hallaoui
A
A
Elachqar
A
A
Lavergne
J-P
JP
Roumestant
M-L
ML
Viallefont
Ph
P
D000596:Amino Acids / Q000737:chemistry*; D004952:Esters; D006571:Heterocyclic Compounds / Q000138:chemical synthesis*; D015394:Molecular Structure
D000596:Amino Acids; D004952:Esters; D006571:Heterocyclic Compounds