Site-specific fluorescent labeling of estrogen receptors and structure-activity relationships of ligands in terms of receptor dimer stability.
Tamrazi
Anobel
A
Department of Chemistry, University of Illinois, Urbana, Illinois 61801-3792, USA.
Katzenellenbogen
John A
JA
D000818:Animals; D001671:Biochemistry / Q000379:methods; D003545:Cysteine / Q000737:chemistry; D019281:Dimerization; D004305:Dose-Response Relationship, Drug; D031541:Fluorescence Resonance Energy Transfer / Q000379:methods; D005456:Fluorescent Dyes / Q000494:pharmacology*; D007700:Kinetics; D008024:Ligands; D010455:Peptides / Q000737:chemistry; D011960:Receptors, Estrogen / Q000737:chemistry*; D013329:Structure-Activity Relationship; D013816:Thermodynamics
D005456:Fluorescent Dyes; D008024:Ligands; D010455:Peptides; D011960:Receptors, Estrogen; D003545:Cysteine