New trifluoromethanesulfonanilide compounds having high miticidal activity against house dust mites.
Several 2-alkoxycarbonyltrifluoromethanesulfonanilides were prepared to examine their miticidal activity. 4-Halo-2-alkoxycarbonyltrifluoromethanesulfonanilides in particular showed good miticidal activity against Tyrophagus putrescentiae (Tp), Dermatophagoides farinae (Dp) and Chelacaropsis moorei (Cm). Amidoflumet (methyl 5-chloro-2-[(trifluoromethyl)sulfonyl]aminobenzoate) was selected and has been developed as a new miticide for house dust mites.
Mori
Tatsuya
T
Agricultural Chemicals Research Laboratory, Sumitomo Chemical Co, Ltd, Takarazuka, Hyogo, Japan. morit7@sc.sumitomo-chem.co.jp
Takada
Yoji
Y
Hatakoshi
Makoto
M
Matsuo
Noritada
N
D000818:Animals; D007202:Indicators and Reagents; D007306:Insecticides / Q000138:chemical synthesis* / Q000494:pharmacology*; D009682:Magnetic Resonance Spectroscopy; D013058:Mass Spectrometry; D008925:Mites / Q000502:physiology*; D013329:Structure-Activity Relationship; D013449:Sulfonamides / Q000138:chemical synthesis* / Q000494:pharmacology*; D062367:ortho-Aminobenzoates / Q000138:chemical synthesis* / Q000494:pharmacology*
D007202:Indicators and Reagents; D007306:Insecticides; D013449:Sulfonamides; D062367:ortho-Aminobenzoates