Strategic Research Institute G-Protein-Coupled Receptors Drug Discovery World Summit.
The Strategic Research Institute provided a well-organised 2-day summit that offered presentations and posters on new assay technology, structure-based small-molecule discovery and examples of clinical candidates targeted to G-protein-coupled receptor (GPCR) targets. A wide variety of topics were presented providing recent advances in GPCR target selection, bioassay-enabling technology and medicinal chemistry targeted to GPCR-relevant chemical libraries. GPCRs continue to be an attractive platform for drug discovery.
Eli Lilly Research Laboratories, Neuroscience Division, Indianapolis, IN, USA. Felder@lilly.com
Christian C
CC
Felder
D000818:Animals; D002626:Chemistry, Pharmaceutical / Q000379:methods; D015195:Drug Design; D015507:Drugs, Investigational / Q000494:pharmacology*; D006801:Humans; D051379:Mice; D043562:Receptors, G-Protein-Coupled / Q000378:metabolism*
D015507:Drugs, Investigational; D043562:Receptors, G-Protein-Coupled