title: Synthesis of novel polycyclic indolyldiamines.
abstract: A rapid and stereoselective access to novel polycyclic indolyldiamines is described. The key step involves simple chemoselective transformations of a common bicyclic aminal intermediate, easily available on a large scale from an enantiomerically pure cyano oxazolopiperidine precursor.
authors.affiliation: Laboratoire de Chimie Thérapeutique, Faculté des Sciences Pharmaceutiques et Biologiques, UMR 8638 associée au CNRS et à l'Université René Descartes, Paris.
authors.forename: Sabrina
authors.initials: S
authors.lastname: Cutri
authors.forename: Anna
authors.initials: A
authors.lastname: Diez
authors.forename: Martine
authors.initials: M
authors.lastname: Bonin
authors.forename: Laurent
authors.initials: L
authors.lastname: Micouin
authors.forename: Henri-Philippe
authors.initials: HP
authors.lastname: Husson