Regio- and chemoselective 6'-N-derivatization of aminoglycosides: bisubstrate inhibitors as probes to study aminoglycoside 6'-N-acetyltransferases.
Gao
Feng
F
Department of Chemistry, McGill University, 801 Sherbrooke Street West, Montréal, Québec, H3A 2K6, Canada.
Yan
Xuxu
X
Baettig
Oliver M
OM
Berghuis
Albert M
AM
Auclair
Karine
K
D000123:Acetyltransferases / Q000138:chemical synthesis / Q000737:chemistry*; D016984:Enterococcus faecium / Q000201:enzymology; D008163:Luminescent Measurements; D011487:Protein Conformation; D017434:Protein Structure, Tertiary; D013237:Stereoisomerism
D000123:Acetyltransferases; C056532:aminoglycoside N(6')-acetyltransferase