title: Structure-activity relationship and pharmacology of gamma-aminobutyric acid (GABA) transport inhibitors.
authors.affiliation: Department of Medicinal Chemistry, The Danish University of Pharmaceutical Sciences, 2 Universitetsparken, DK-2100 Copenhagen, Denmark.
authors.forename: Rasmus Praetorius
authors.initials: RP
authors.lastname: Clausen
authors.forename: Karsten
authors.initials: K
authors.lastname: Madsen
authors.forename: Orla Miller
authors.initials: OM
authors.lastname: Larsson
authors.forename: Bente
authors.initials: B
authors.lastname: Frølund
authors.forename: Povl
authors.initials: P
authors.lastname: Krogsgaard-Larsen
authors.forename: Arne
authors.initials: A
authors.lastname: Schousboe
mesh_terms: D000818:Animals; D018755:GABA Agonists / Q000737:chemistry / Q000494:pharmacology; D018756:GABA Antagonists / Q000737:chemistry / Q000494:pharmacology; D050485:GABA Plasma Membrane Transport Proteins / Q000378:metabolism; D058805:GABA Uptake Inhibitors; D006801:Humans; D015394:Molecular Structure; D014179:Neurotransmitter Uptake Inhibitors / Q000737:chemistry / Q000494:pharmacology*; D009557:Nipecotic Acids / Q000737:chemistry / Q000494:pharmacology; D010091:Oximes / Q000737:chemistry / Q000494:pharmacology; D013329:Structure-Activity Relationship; D000078308:Tiagabine
chemical_list: D018755:GABA Agonists; D018756:GABA Antagonists; D050485:GABA Plasma Membrane Transport Proteins; D058805:GABA Uptake Inhibitors; D014179:Neurotransmitter Uptake Inhibitors; D009557:Nipecotic Acids; D010091:Oximes; C078793:NNC 711; D000078308:Tiagabine