Synthesis of insecticidal fluorinated anthranilic diamides.
A series of highly active fluorinated anthranilic diamide insecticides have been prepared and their biological activity assessed on two aphid species in the search for systemically active compounds that control Hemiptera. In addition, we have demonstrated a new synthesis of N-aryl 3-fluoropyrazoles.
Clark
David A
DA
DuPont Crop Protection, Stine-Haskell Research Center, PO Box 30, Newark, DE 19714, USA. david.a.clark@usa.dupont.com
Lahm
George P
GP
Smith
Ben K
BK
Barry
James D
JD
Clagg
Don G
DG
D000577:Amides / Q000737:chemistry / Q000494:pharmacology; D000818:Animals; D001042:Aphids / Q000187:drug effects*; D054879:Halogenation; D006430:Hemiptera / Q000187:drug effects; D007306:Insecticides / Q000138:chemical synthesis*; D011720:Pyrazoles; D062367:ortho-Aminobenzoates / Q000737:chemistry* / Q000494:pharmacology*
D000577:Amides; D007306:Insecticides; D011720:Pyrazoles; D062367:ortho-Aminobenzoates