A tandem elimination-cyclization-Suzuki approach: efficient one-pot synthesis of functionalized (Z)-3-(arylmethylene)isoindolin-1-ones.
A novel and efficient one-pot regioselective elimination-cyclization-Suzuki approach was developed to afford (Z)-3-arylmethyleneisoindolin-1-ones in good to excellent yields from easily accessible o-gem-dihalovinylbenzamides and organoboron reagents.
Sun
Caiyun
C
Department of Chemistry, Shanghai University, Shanghai 200444, China.
Xu
Bin
B
D001549:Benzamides / Q000138:chemical synthesis / Q000737:chemistry; D001896:Boron Compounds / Q000737:chemistry; D003500:Cyclization; D007211:Indoles / Q000138:chemical synthesis* / Q000737:chemistry; D015394:Molecular Structure; D013237:Stereoisomerism
D001549:Benzamides; D001896:Boron Compounds; D007211:Indoles