Microwave-assisted Suzuki-Miyaura couplings on α-iodoenaminones.
A systematic study of α-iodination and subsequent Suzuki-Miyaura couplings between non-attenuated enaminones and a wide range of aromatic boronic acids is reported. The microwave-assisted variant of this transformation furnished the α-arylenaminones in significantly shorter reaction times and slightly improved yields as compared to conventional heating.
Wang
Xin
X
Department of Medicinal Chemistry and Center for Methodology and Library Development, University of Kansas, 1251 Wescoe Hall Drive, Lawrence, Kansas 66045, USA.
Turunen
Brandon J
BJ
Leighty
Matthew W
MW
Georg
Gunda I
GI