title: N-->S acyl-transfer-mediated synthesis of peptide thioesters using anilide derivatives.
abstract: N-->S acyl-transfer-mediated synthesis of peptide thioesters utilizing an N-aminoacyl-N-sulfanylethylaminobenzoic acid derivative has been examined. The developed synthetic methodology for peptide thioesters is compatible with Fmoc solid-phase peptide synthesis (SPPS).
authors.affiliation: Institute of Health Biosciences and Graduate School of Pharmaceutical Sciences, The University of Tokushima, Tokushima 770-8505, Japan.
authors.forename: Shugo
authors.initials: S
authors.lastname: Tsuda
authors.forename: Akira
authors.initials: A
authors.lastname: Shigenaga
authors.forename: Kiyomi
authors.initials: K
authors.lastname: Bando
authors.forename: Akira
authors.initials: A
authors.lastname: Otaka
mesh_terms: D000813:Anilides / Q000737:chemistry*; D004952:Esters; D015394:Molecular Structure; D009584:Nitrogen / Q000737:chemistry; D010455:Peptides / Q000138:chemical synthesis* / Q000737:chemistry; D013455:Sulfur / Q000737:chemistry
chemical_list: D000813:Anilides; D004952:Esters; D010455:Peptides; D013455:Sulfur; D009584:Nitrogen