Design, synthesis, and biological activities of novel 2-cyanoacrylates containing oxazole, oxadiazole, or quinoline moieties.
A series of novel 2-cyanoacrylates containing an oxazole, oxadiazole, or quinoline moiety were designed and synthesized, and their structures were characterized by (1)H NMR and elemental analysis (or high-resolution mass spectrometry). Their herbicidal activities against four weeds were evaluated, and the result indicated that some of the title compounds showed excellent herbicidal activities against rape and amaranth pigweed in postemergence treatment at a dose of 375 g/ha. Furthermore, most of these cyanoacrylates exhibited interesting plant growth regulatory activities.
Zhao
Qiqi
Q
State Key Laboratory of Elemento-Organic Chemistry, Research Institute of Elemento-Organic Chemistry, Nankai University, Tianjin 300071, People's Republic of China.
Liu
Shaohua
S
Li
Yonghong
Y
Wang
Qingmin
Q
D027721:Amaranthus / Q000187:drug effects; D029688:Brassica napus / Q000187:drug effects; D031746:Digitaria / Q000187:drug effects; D015195:Drug Design; D004659:Enbucrilate / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D006540:Herbicides / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology; D009682:Magnetic Resonance Spectroscopy; D000455:Medicago sativa / Q000187:drug effects; D010069:Oxadiazoles / Q000032:analysis*; D010080:Oxazoles / Q000032:analysis*; D045332:Photosystem II Protein Complex / Q000037:antagonists & inhibitors; D010937:Plant Growth Regulators / Q000494:pharmacology; D011804:Quinolines / Q000032:analysis*
D006540:Herbicides; D010069:Oxadiazoles; D010080:Oxazoles; D045332:Photosystem II Protein Complex; D010937:Plant Growth Regulators; D011804:Quinolines; D004659:Enbucrilate