Expedient and rapid synthesis of 1,2,3-triazolo[5,1-c]morpholines through palladium-copper catalysis.
A one-pot approach using palladium-copper as catalyst has been developed for the synthesis of morpholines fused with 1,2,3-triazole. Good regioselectivity, mild reaction conditions, high yields and short reaction time are the hallmarks of this method.
Chowdhury
Chinmay
C
Chemistry Division, Indian Institute of Chemical Biology (unit of CSIR), 4, Raja S. C. Mullick Road, Jadavpur, Kolkata 700032, India. chinmay@iicb.res.in
Mukherjee
Sanjukta
S
Das
Bimolendu
B
Achari
Basudeb
B