The synthesis of DAMGO-based potential affinity labels with high mu opioid receptor affinity and the formation of cyclic O-alkyl thiocarbamates.
Dattachowdhury
Bhaswati
B
Department of Medicinal Chemistry, University of Kansas, Lawrence, KS 66045, USA.
Murray
Thomas F
TF
Aldrich
Jane V
JV
D000345:Affinity Labels; D020875:Enkephalin, Ala(2)-MePhe(4)-Gly(5)- / Q000138:chemical synthesis*; D009682:Magnetic Resonance Spectroscopy; D017450:Receptors, Opioid, mu / Q000378:metabolism*; D013859:Thiocarbamates / Q000378:metabolism*
D000345:Affinity Labels; D017450:Receptors, Opioid, mu; D013859:Thiocarbamates; D020875:Enkephalin, Ala(2)-MePhe(4)-Gly(5)-