Enantioselective aza-Darzens reaction catalyzed by a chiral phosphoric acid.
Aza-Darzens reaction of ethyl diazoacetate with aldimines, derived from phenyl glyoxal, furnished cis-aziridine carboxylates with excellent enantioselectivities by means of a chiral phosphoric acid.
Akiyama
Takahiko
T
Department of Chemistry, Gakushuin University, 1-5-1 Mejiro, Toshima-ku, Tokyo 171-8588, Japan. takahiko.akiyama@gakushuin.ac.jp
Suzuki
Tohru
T
Mori
Keiji
K