title: Through the "gatekeeper door": exploiting the active kinase conformation.
authors.affiliation: Department of Chemical Core Technologies, Nerviano Medical Sciences, Oncology, Viale Pasteur 10, Nerviano 20014, Italy. Fabio.Zuccotto@Nervianoms.com
authors.forename: Fabio
authors.initials: F
authors.lastname: Zuccotto
authors.forename: Elena
authors.initials: E
authors.lastname: Ardini
authors.forename: Elena
authors.initials: E
authors.lastname: Casale
authors.forename: Mauro
authors.initials: M
authors.lastname: Angiolini
mesh_terms: D015195:Drug Design; D006801:Humans; D047428:Protein Kinase Inhibitors / Q000737:chemistry / Q000494:pharmacology; D011494:Protein Kinases / Q000737:chemistry* / Q000378:metabolism*; D013379:Substrate Specificity
chemical_list: D047428:Protein Kinase Inhibitors; D011494:Protein Kinases