Palladium-catalyzed tandem amination reaction for the synthesis of 4-quinolones.
An efficient palladium-catalyzed tandem amination approach was developed in one step to afford functionalized 4-quinolones in good to excellent yields from easily accessible o-haloaryl acetylenic ketones and primary amines.
Zhao
Tiankun
T
Department of Chemistry, Shanghai University, Shanghai 200444, China.
Xu
Bin
B
D042462:4-Quinolones / Q000138:chemical synthesis* / Q000737:chemistry; D000586:Amination; D000588:Amines / Q000737:chemistry; D002384:Catalysis; D007659:Ketones / Q000737:chemistry; D015394:Molecular Structure; D010165:Palladium / Q000737:chemistry*
D042462:4-Quinolones; D000588:Amines; D007659:Ketones; D010165:Palladium