title: Phenyl-oxazoles, a new family of inverse agonists at the H(3) histamine receptor.
authors.affiliation: UCB New Medicines, Chemin du Foriest, 1420 Braine-L'Alleud, Belgium. Frederic.denonne@ucb.com
authors.forename: Frédéric
authors.initials: F
authors.lastname: Denonne
authors.forename: Franck
authors.initials: F
authors.lastname: Atienzar
authors.forename: Sylvain
authors.initials: S
authors.lastname: Célanire
authors.forename: Bernard
authors.initials: B
authors.lastname: Christophe
authors.forename: Frédérique
authors.initials: F
authors.lastname: Delannois
authors.forename: Christel
authors.initials: C
authors.lastname: Delaunoy
authors.forename: Marie-Laure
authors.initials: ML
authors.lastname: Delporte
authors.forename: Véronique
authors.initials: V
authors.lastname: Durieu
authors.forename: Michel
authors.initials: M
authors.lastname: Gillard
authors.forename: Bénédicte
authors.initials: B
authors.lastname: Lallemand
authors.forename: Yves
authors.initials: Y
authors.lastname: Lamberty
authors.forename: Geneviève
authors.initials: G
authors.lastname: Lorent
authors.forename: Alain
authors.initials: A
authors.lastname: Vanbellinghen
authors.forename: Nathalie
authors.initials: N
authors.lastname: Van Houtvin
authors.forename: Valérie
authors.initials: V
authors.lastname: Verbois
authors.forename: Laurent
authors.initials: L
authors.lastname: Provins
mesh_terms: D000818:Animals; D001554:Benzene / Q000737:chemistry*; D018938:Caco-2 Cells; D002460:Cell Line; D003072:Cognition Disorders / Q000188:drug therapy; D054314:Drug Inverse Agonism; D006633:Histamine Antagonists / Q000737:chemistry*; D006801:Humans; D008297:Male; D051379:Mice; D008862:Microsomes, Liver / Q000378:metabolism; D010080:Oxazoles / Q000737:chemistry* / Q000493:pharmacokinetics; D011759:Pyrrolidines / Q000737:chemistry* / Q000493:pharmacokinetics; D051381:Rats; D017207:Rats, Sprague-Dawley; D018100:Receptors, Histamine H3 / Q000737:chemistry* / Q000378:metabolism; D013329:Structure-Activity Relationship; D013844:Thiazoles / Q000737:chemistry / Q000493:pharmacokinetics
chemical_list: D006633:Histamine Antagonists; D010080:Oxazoles; D011759:Pyrrolidines; D018100:Receptors, Histamine H3; D013844:Thiazoles; D001554:Benzene