Identification of potent, highly constrained CGRP receptor antagonists.
Stump
Craig A
CA
Department of Medicinal Chemistry, Merck & Co., Inc., West Point, PA 19486, USA. craig_stump@merck.com
Bell
Ian M
IM
Bednar
Rodney A
RA
Fay
John F
JF
Gallicchio
Steven N
SN
Hershey
James C
JC
Jelley
Richard
R
Kreatsoulas
Constantine
C
Moore
Eric L
EL
Mosser
Scott D
SD
Quigley
Amy G
AG
Roller
Shane A
SA
Salvatore
Christopher A
CA
Sharik
Steven S
SS
Theberge
Cory R
CR
Zartman
C Blair
CB
Kane
Stefanie A
SA
Graham
Samuel L
SL
Selnick
Harold G
HG
Vacca
Joseph P
JP
Williams
Theresa M
TM
D000818:Animals; D001682:Biological Availability; D000077221:Calcitonin Gene-Related Peptide Receptor Antagonists; D004285:Dogs; D004353:Drug Evaluation, Preclinical; D008253:Macaca mulatta; D011804:Quinolines / Q000737:chemistry / Q000493:pharmacokinetics / Q000494:pharmacology*; D051381:Rats
D000077221:Calcitonin Gene-Related Peptide Receptor Antagonists; D011804:Quinolines