Radioligand binding characterization of the bradykinin B(2) receptor in the rabbit and pig ileal smooth muscle.
Meini
Stefania
S
Department of Pharmacology, Menarini Ricerche S.p.A., via Rismondo 12A, Florence, Italy. smeini@menarini-ricerche.it
Cucchi
Paola
P
Catalani
Claudio
C
Bellucci
Francesca
F
Santicioli
Paolo
P
Giuliani
Sandro
S
Maggi
Carlo Alberto
CA
D000818:Animals; D001920:Bradykinin / Q000378:metabolism; D065094:Bradykinin B2 Receptor Antagonists; D002462:Cell Membrane / Q000378:metabolism; D005260:Female; D006168:Guinea Pigs; D006801:Humans; D007082:Ileum; D008024:Ligands; D008297:Male; D051379:Mice; D009130:Muscle, Smooth / Q000166:cytology / Q000378:metabolism*; D009952:Ornithine / Q000031:analogs & derivatives / Q000378:metabolism / Q000494:pharmacology; D011485:Protein Binding / Q000187:drug effects; D011817:Rabbits; D043782:Receptor, Bradykinin B2 / Q000378:metabolism*; D013379:Substrate Specificity; D013449:Sulfonamides / Q000378:metabolism / Q000494:pharmacology; D013552:Swine
C506838:(4-amino-5-(4-(4-(2,4-dichloro-3-(2,4-dimethyl-8-quinolyloxymethyl)phenylsulfonamido)tetrahydro-2H-4-pyranoylcarbonyl)piperazino)-5-oxopentyl)(trimethyl)ammonium; D065094:Bradykinin B2 Receptor Antagonists; D008024:Ligands; D043782:Receptor, Bradykinin B2; D013449:Sulfonamides; D009952:Ornithine; D001920:Bradykinin