20S proteasome inhibition: designing noncovalent linear peptide mimics of the natural product TMC-95A.
Groll
Michael
M
Department Chemie, Lehrstuhl für Biochemie, Technische Universität München, Garching Germany. michael.groll@ch.tum.de
Gallastegui
Nerea
N
Maréchal
Xavier
X
Le Ravalec
Virginie
V
Basse
Nicolas
N
Richy
Nicolas
N
Genin
Emilie
E
Huber
Robert
R
Moroder
Luis
L
Vidal
Joëlle
J
Reboud-Ravaux
Michèle
M
D001665:Binding Sites; D020134:Catalytic Domain; D018360:Crystallography, X-Ray; D010456:Peptides, Cyclic / Q000737:chemistry* / Q000494:pharmacology; D011480:Protease Inhibitors / Q000737:chemistry* / Q000494:pharmacology; D046988:Proteasome Endopeptidase Complex / Q000378:metabolism; D061988:Proteasome Inhibitors
D010456:Peptides, Cyclic; D011480:Protease Inhibitors; D061988:Proteasome Inhibitors; C408291:TMC-95A; D046988:Proteasome Endopeptidase Complex