Development of Practical Methodologies for the Synthesis of Functionalized Benzoboroxoles.
2-Formylphenylboronic acids upon reaction with activated olefins such as acrylates, methyl vinyl ketone, and acrylonitrile, etc. provide functionalized benzoboroxoles. The corresponding homologated benzoboroxoles were synthesized via the reaction of 2-formylphenylboronic acids with α-bromomethylacrylates.
Kumar
J Sravan
JS
Department of Chemistry and Biochemistry, University of Minnesota Duluth, Duluth, MN 55812.
Bashian
Christopher M
CM
Corsello
Michael A
MA
Jonnalagadda
Subash C
SC
Mereddy
Venkatram R
VR
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