Aminopyrazine inhibitors binding to an unusual inactive conformation of the mitotic kinase Nek2: SAR and structural characterization.
Whelligan
Daniel K
DK
Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research, 15 Cotswold Road, Sutton, Surrey SM2 5NG, United Kingdom.
Solanki
Savade
S
Taylor
Dawn
D
Thomson
Douglas W
DW
Cheung
Kwai-Ming J
KM
Boxall
Kathy
K
Mas-Droux
Corine
C
Barillari
Caterina
C
Burns
Samantha
S
Grummitt
Charles G
CG
Collins
Ian
I
van Montfort
Rob L M
RL
Aherne
G Wynne
GW
Bayliss
Richard
R
Hoelder
Swen
S