Development of novel bisubstrate-type inhibitors of histone methyltransferase SET7/9.
Mori
Shuichi
S
Tokyo Medical and Dental University, Chiyoda-ku, Japan.
Iwase
Kenta
K
Iwanami
Naoko
N
Tanaka
Yujiro
Y
Kagechika
Hiroyuki
H
Hirano
Tomoya
T
D004791:Enzyme Inhibitors / Q000138:chemical synthesis / Q000737:chemistry* / Q000494:pharmacology; D011495:Histone-Lysine N-Methyltransferase / Q000037:antagonists & inhibitors* / Q000378:metabolism; D012436:S-Adenosylmethionine / Q000138:chemical synthesis / Q000737:chemistry* / Q000494:pharmacology; D013379:Substrate Specificity
D004791:Enzyme Inhibitors; D012436:S-Adenosylmethionine; D011495:Histone-Lysine N-Methyltransferase; C540312:SETD7 protein, human