title: New cathepsin inhibitors to explore the fluorophilic properties of the S2 pocket of cathepsin B: design, synthesis, and biological evaluation.
authors: Departamento de Química Orgánica, Universidad de Valencia, 46100 Burjassot, Spain. santos.fustero@uv.es
authors: Santos
authors: S
authors: Fustero
authors: Vanessa
authors: V
authors: Rodrigo
authors: María
authors: M
authors: Sánchez-Roselló
authors: Carlos
authors: C
authors: del Pozo
authors: Joaquín
authors: J
authors: Timoneda
authors: Maxim
authors: M
authors: Frizler
authors: Mihiret T
authors: MT
authors: Sisay
authors: Jürgen
authors: J
authors: Bajorath
authors: Luis P
authors: LP
authors: Calle
authors: F Javier
authors: FJ
authors: Cañada
authors: Jesús
authors: J
authors: Jiménez-Barbero
authors: Michael
authors: M
authors: Gütschow
mesh_terms: D002401:Cathepsin B / Q000037:antagonists & inhibitors*; D020650:Combinatorial Chemistry Techniques; D004151:Dipeptides / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D015195:Drug Design; D006801:Humans; D006845:Hydrocarbons, Fluorinated / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D015394:Molecular Structure; D009570:Nitriles / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D013237:Stereoisomerism
chemical_list: D004151:Dipeptides; D006845:Hydrocarbons, Fluorinated; D009570:Nitriles; D002401:Cathepsin B