title: Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G.
abstract: 3-(Hetero)aryl substituted indoles, 7-azaindoles, and pyrroles can be obtained in a very concise fashion via a one-pot Masuda borylation-Suzuki coupling sequence. The concise total syntheses of the marine natural products meridianins A (5) and G (4i) nicely illustrate the utility of this methodology.
authors: Lehrstuhl für Organische Chemie, Institut für Organische Chemie und Makromolekulare Chemie, Heinrich-Heine-Universität Düsseldorf, Universitätsstraße 1, D-40225, Düsseldorf, Germany.
authors: Eugen
authors: E
authors: Merkul
authors: Elisabeth
authors: E
authors: Schäfer
authors: Thomas J J
authors: TJ
authors: Müller
mesh_terms: D001895:Boron / Q000737:chemistry*; D026121:Indole Alkaloids / Q000138:chemical synthesis*; D015394:Molecular Structure; D013997:Time Factors
chemical_list: D026121:Indole Alkaloids; C560347:meridianin A; C522699:meridianin G; D001895:Boron