title: Synthesis of a biologically active triazole-containing analogue of cystatin A through successive peptidomimetic alkyne-azide ligations.
authors.affiliation: Centre de Biophysique Moléculaire, CNRS UPR 4301, Rue Charles Sadron, 45071 Orléans cedex 2, France.
authors.forename: Ibai E
authors.initials: IE
authors.lastname: Valverde
authors.forename: Fabien
authors.initials: F
authors.lastname: Lecaille
authors.forename: Gilles
authors.initials: G
authors.lastname: Lalmanach
authors.forename: Vincent
authors.initials: V
authors.lastname: Aucagne
authors.forename: Agnès F
authors.initials: AF
authors.lastname: Delmas
mesh_terms: D000480:Alkynes / Q000737:chemistry; D000595:Amino Acid Sequence; D001386:Azides / Q000737:chemistry; D002403:Cathepsins / Q000037:antagonists & inhibitors; D045744:Cell Line, Tumor; D057930:Click Chemistry / Q000379:methods*; D003500:Cyclization; D055312:Cystatin A / Q000138:chemical synthesis* / Q000737:chemistry / Q000494:pharmacology*; D006801:Humans; D008969:Molecular Sequence Data; D009361:Neoplasm Invasiveness / Q000517:prevention & control; D057786:Peptidomimetics / Q000737:chemistry*; D014230:Triazoles / Q000138:chemical synthesis / Q000737:chemistry*
chemical_list: D000480:Alkynes; D001386:Azides; D055312:Cystatin A; D057786:Peptidomimetics; D014230:Triazoles; D002403:Cathepsins