title: The dopamine stabilizers ACR16 and (-)-OSU6162 display nanomolar affinities at the σ-1 receptor.
authors.forename: K
authors.initials: K
authors.lastname: Sahlholm
authors.forename: P
authors.initials: P
authors.lastname: Århem
authors.forename: K
authors.initials: K
authors.lastname: Fuxe
authors.forename: D
authors.initials: D
authors.lastname: Marcellino
mesh_terms: D000661:Amphetamine / Q000494:pharmacology; D000818:Animals; D015259:Dopamine Agents / Q000494:pharmacology*; D004305:Dose-Response Relationship, Drug; D004347:Drug Interactions; D057809:HEK293 Cells; D006801:Humans; D008297:Male; D010880:Piperidines / Q000493:pharmacokinetics*; D011485:Protein Binding / Q000187:drug effects; D011869:Radioligand Assay / Q000379:methods; D051381:Rats; D017207:Rats, Sprague-Dawley; D017480:Receptors, sigma / Q000235:genetics / Q000378:metabolism*; D014162:Transfection; D014316:Tritium / Q000493:pharmacokinetics; D000097605:Sigma-1 Receptor
chemical_list: D000661:Amphetamine; D015259:Dopamine Agents; D010880:Piperidines; D017480:Receptors, sigma; D014316:Tritium; D000097605:Sigma-1 Receptor; C109513:OSU 6162; C483720:pridopidine