title: Azetidine iminosugars from the cyclization of 3,5-di-O-triflates of α-furanosides and of 2,4-di-O-triflates of β-pyranosides derived from glucose.
abstract: Primary amines with either 3,5-di-O-ditriflates of α-furanosides or 2,4-di-O-triflates of β-pyranosides form bicyclic azetidines in high yield.
authors.affiliation: Chemistry Research Laboratory, Department of Chemistry, University of Oxford, Mansfield Road, Oxford, OX1 3TA, UK.
authors.forename: Gabriel M J
authors.initials: GM
authors.lastname: Lenagh-Snow
authors.forename: Noelia
authors.initials: N
authors.lastname: Araújo
authors.forename: Sarah F
authors.initials: SF
authors.lastname: Jenkinson
authors.forename: R Fernando
authors.initials: RF
authors.lastname: Martínez
authors.forename: Yousuke
authors.initials: Y
authors.lastname: Shimada
authors.forename: Chu-Yi
authors.initials: CY
authors.lastname: Yu
authors.forename: Atsushi
authors.initials: A
authors.lastname: Kato
authors.forename: George W J
authors.initials: GW
authors.lastname: Fleet
mesh_terms: D000588:Amines / Q000737:chemistry*; D001384:Azetidines / Q000138:chemical synthesis* / Q000737:chemistry; D003500:Cyclization; D005947:Glucose / Q000737:chemistry*; D050111:Imino Sugars / Q000138:chemical synthesis* / Q000737:chemistry; D008698:Mesylates / Q000737:chemistry*; D015394:Molecular Structure; D013329:Structure-Activity Relationship
chemical_list: D000588:Amines; D001384:Azetidines; D050111:Imino Sugars; D008698:Mesylates; D005947:Glucose