title: 6-halogenochromones bearing tryptamine: one-step access to potent and highly selective inhibitors of breast cancer resistance protein.
authors.affiliation: Mechanisms and Modulation of Drug Resistance Team, Institute of Biology and Chemistry of Proteins, BMSSI UMR 5086 CNRS/University of Lyon 1, 7 Passage du Vercors, 69367 Lyon, France.
authors.forename: Glaucio
authors.initials: G
authors.lastname: Valdameri
authors.forename: Estelle
authors.initials: E
authors.lastname: Genoux-Bastide
authors.forename: Charlotte
authors.initials: C
authors.lastname: Gauthier
authors.forename: Basile
authors.initials: B
authors.lastname: Peres
authors.forename: Raphaël
authors.initials: R
authors.lastname: Terreux
authors.forename: Sheila M B
authors.initials: SM
authors.lastname: Winnischofer
authors.forename: Maria E M
authors.initials: ME
authors.lastname: Rocha
authors.forename: Attilio
authors.initials: A
authors.lastname: Di Pietro
authors.forename: Ahcène
authors.initials: A
authors.lastname: Boumendjel
mesh_terms: D000070997:ATP Binding Cassette Transporter, Subfamily G, Member 2; D018528:ATP-Binding Cassette Transporters / Q000037:antagonists & inhibitors* / Q000378:metabolism; D000970:Antineoplastic Agents / Q000138:chemical synthesis / Q000737:chemistry / Q000494:pharmacology*; D049109:Cell Proliferation / Q000187:drug effects; D002470:Cell Survival / Q000187:drug effects; D002478:Cells, Cultured; D002867:Chromones / Q000138:chemical synthesis / Q000737:chemistry / Q000494:pharmacology*; D004305:Dose-Response Relationship, Drug; D004354:Drug Screening Assays, Antitumor; D057809:HEK293 Cells; D006801:Humans; D015394:Molecular Structure; D009363:Neoplasm Proteins / Q000037:antagonists & inhibitors* / Q000378:metabolism; D013329:Structure-Activity Relationship; D014363:Tryptamines / Q000737:chemistry*
chemical_list: C116614:ABCG2 protein, human; D000070997:ATP Binding Cassette Transporter, Subfamily G, Member 2; D018528:ATP-Binding Cassette Transporters; D000970:Antineoplastic Agents; D002867:Chromones; D009363:Neoplasm Proteins; D014363:Tryptamines; C030820:tryptamine