title: Copper-catalyzed ortho-halogenation of protected anilines.
abstract: A practical Cu-catalyzed direct ortho-halogenation of anilines under aerobic conditions has been developed. The reaction shows typically excellent mono-substitution selectivity, high ortho-regiocontrol and large functional group tolerance.
authors.affiliation: Departamento de Química Orgánica, Universidad Autónoma de Madrid, Cantoblanco, 28049 Madrid, Spain. n.rodriguez@uam.es ramon.gomez@uam.es juancarlos.carretero@uam.es.
authors.forename: Beatriz
authors.initials: B
authors.lastname: Urones
authors.forename: Ángel Manu
authors.initials: ÁM
authors.lastname: Martínez
authors.forename: Nuria
authors.initials: N
authors.lastname: Rodríguez
authors.forename: Ramón Gómez
authors.initials: RG
authors.lastname: Arrayás
authors.forename: Juan C
authors.initials: JC
authors.lastname: Carretero