title: Vicinal disulfide constrained cyclic peptidomimetics: a turn mimetic scaffold targeting the norepinephrine transporter.
authors.affiliation: Institute of Molecular Bioscience, The University of Queensland, St Lucia QLD 4072 (Australia). a.brust@imb.uq.edu.au.
authors.forename: Andreas
authors.initials: A
authors.lastname: Brust
authors.forename: Ching-I A
authors.initials: CI
authors.lastname: Wang
authors.forename: Norelle L
authors.initials: NL
authors.lastname: Daly
authors.forename: Joseph
authors.initials: J
authors.lastname: Kennerley
authors.forename: Mahsa
authors.initials: M
authors.lastname: Sadeghi
authors.forename: Macdonald J
authors.initials: MJ
authors.lastname: Christie
authors.forename: Richard J
authors.initials: RJ
authors.lastname: Lewis
authors.forename: Mehdi
authors.initials: M
authors.lastname: Mobli
authors.forename: Paul F
authors.initials: PF
authors.lastname: Alewood
mesh_terms: D018759:Adrenergic Uptake Inhibitors / Q000097:blood / Q000138:chemical synthesis / Q000737:chemistry; D000595:Amino Acid Sequence; D000818:Animals; D004220:Disulfides / Q000737:chemistry*; D004353:Drug Evaluation, Preclinical; D006207:Half-Life; D006801:Humans; D009682:Magnetic Resonance Spectroscopy; D050484:Norepinephrine Plasma Membrane Transport Proteins / Q000037:antagonists & inhibitors* / Q000378:metabolism; D010456:Peptides, Cyclic / Q000097:blood / Q000138:chemical synthesis / Q000737:chemistry; D057786:Peptidomimetics; D017434:Protein Structure, Tertiary; D051381:Rats
chemical_list: D018759:Adrenergic Uptake Inhibitors; D004220:Disulfides; D050484:Norepinephrine Plasma Membrane Transport Proteins; D010456:Peptides, Cyclic; D057786:Peptidomimetics
keywords: biological activity; combinatorial chemistry; cyclic peptides; drug discovery; peptidomimetics