title: Copper-catalyzed sequential N-arylation of C-amino-NH-azoles.
abstract: Copper(II)-catalyzed boronic acid promoted C-N bond cross-coupling reactions have been successfully developed for sequential N-arylation of C-amino-NH-azoles. These general protocols are compatible with a variety of aryl/hetero-aryl boronic acids and provided rapid access to a diverse array of diarylaminoazole derivatives in a two-step sequence or in one-pot.
authors.affiliation: Academy of Scientific and Innovative Research (AcSIR), Canal Road, Jammu-180001, India.
authors.forename: D Nageswar
authors.initials: DN
authors.lastname: Rao
authors.forename: Sk
authors.initials: S
authors.lastname: Rasheed
authors.forename: Ram A
authors.initials: RA
authors.lastname: Vishwakarma
authors.forename: Parthasarathi
authors.initials: P
authors.lastname: Das
mesh_terms: D000586:Amination; D001393:Azoles / Q000138:chemical synthesis* / Q000737:chemistry; D001897:Boronic Acids / Q000737:chemistry*; D002384:Catalysis; D003300:Copper / Q000737:chemistry*; D006841:Hydrocarbons, Aromatic / Q000737:chemistry*
chemical_list: D001393:Azoles; D001897:Boronic Acids; D006841:Hydrocarbons, Aromatic; D003300:Copper