title: Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles.
abstract: A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.
authors.affiliation: Department Chemie and Catalysis Research Center (CRC), Technische Universität München, 85747 Garching, Germany. thorsten.bach@ch.tum.de.
authors.forename: Julian
authors.initials: J
authors.lastname: Wippich
authors.forename: Ingo
authors.initials: I
authors.lastname: Schnapperelle
authors.forename: Thorsten
authors.initials: T
authors.lastname: Bach