title: Selective remote C-H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis.
abstract: Copper-catalysed direct C-H bond sulfonylation of aminoquinolines using commercially available and inexpensive arylsulfonyl chlorides as the sulfonylation reagents is described. The reactions took place exclusively at the C5-H position of the quinoline rings and tolerated a wide spectrum of functional groups. Moreover, synthetic transformations of the sulfonylated products led to useful compounds.
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Hong-Wen
authors.initials: HW
authors.lastname: Liang
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Kun
authors.initials: K
authors.lastname: Jiang
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Wei
authors.initials: W
authors.lastname: Ding
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Yi
authors.initials: Y
authors.lastname: Yuan
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Li
authors.initials: L
authors.lastname: Shuai
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Ying-Chun
authors.initials: YC
authors.lastname: Chen
authors.affiliation: College of Pharmacy, Third Military Medical University, Chongqing 400038, China. weiye712@hotmail.com.
authors.forename: Ye
authors.initials: Y
authors.lastname: Wei