Discovery of Chemical Inhibitors of Human Bromodomains.
Department of Structural and Chemical Biology, Icahn School of Medicine at Mount Sinai , 1425 Madison Avenue, New York, New York 10029, United States.
Guangtao
G
Zhang
Department of Structural and Chemical Biology, Icahn School of Medicine at Mount Sinai , 1425 Madison Avenue, New York, New York 10029, United States.
Steven G
SG
Smith
Department of Structural and Chemical Biology, Icahn School of Medicine at Mount Sinai , 1425 Madison Avenue, New York, New York 10029, United States.
Ming-Ming
MM
Zhou
D000123:Acetyltransferases / Q000037:antagonists & inhibitors* / Q000378:metabolism; D001381:Azepines / Q000737:chemistry / Q000378:metabolism; D001391:Azo Compounds / Q000737:chemistry / Q000378:metabolism; D002227:Carbazoles / Q000737:chemistry / Q000378:metabolism; D003959:Diamines / Q000737:chemistry / Q000378:metabolism; D004353:Drug Evaluation, Preclinical; D006801:Humans; D011485:Protein Binding; D017434:Protein Structure, Tertiary; D011804:Quinolines / Q000737:chemistry / Q000378:metabolism; D054852:Small Molecule Libraries / Q000737:chemistry / Q000378:metabolism*; D014157:Transcription Factors / Q000037:antagonists & inhibitors* / Q000378:metabolism
D001381:Azepines; D001391:Azo Compounds; D002227:Carbazoles; D003959:Diamines; D011804:Quinolines; D054852:Small Molecule Libraries; D014157:Transcription Factors; D000123:Acetyltransferases