title: Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines.
abstract: Cu-catalyzed three-component couplings of vinylazaarenes, B2(pin)2, and N-Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities.
authors.affiliation: EaStCHEM, School of Chemistry, University of Edinburgh, Joseph Black Building, The King's Buildings, David Brewster Road, Edinburgh, EH9 3FJ, UK and School of Chemistry, University of Nottingham, University Park, Nottingham, NG7 2RD, UK. hon.lam@nottingham.ac.uk.
authors.forename: Joshua J
authors.initials: JJ
authors.lastname: Smith
authors.affiliation: EaStCHEM, School of Chemistry, University of Edinburgh, Joseph Black Building, The King's Buildings, David Brewster Road, Edinburgh, EH9 3FJ, UK and School of Chemistry, University of Nottingham, University Park, Nottingham, NG7 2RD, UK. hon.lam@nottingham.ac.uk.
authors.forename: Daniel
authors.initials: D
authors.lastname: Best
authors.affiliation: EaStCHEM, School of Chemistry, University of Edinburgh, Joseph Black Building, The King's Buildings, David Brewster Road, Edinburgh, EH9 3FJ, UK and School of Chemistry, University of Nottingham, University Park, Nottingham, NG7 2RD, UK. hon.lam@nottingham.ac.uk.
authors.forename: Hon Wai
authors.initials: HW
authors.lastname: Lam