title: Regioselective Ir(III)-catalyzed C-H alkynylation directed by 7-azaindoles.
abstract: Herein we report a novel iridium(iii)-catalyzed ortho-mono-alkynylation of 7-azaindoles under mild conditions. This approach provides a general and straightforward access to form novel 7-azaindole derivatives with ample substrate scope and broad group tolerance.
authors.affiliation: Skate Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, China. lirt@bjmu.edu.cn.
authors.forename: Bin
authors.initials: B
authors.lastname: Liu
authors.affiliation: Skate Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, China. lirt@bjmu.edu.cn.
authors.forename: Xin
authors.initials: X
authors.lastname: Wang
authors.affiliation: Skate Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, China. lirt@bjmu.edu.cn.
authors.forename: Zemei
authors.initials: Z
authors.lastname: Ge
authors.affiliation: Skate Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, China. lirt@bjmu.edu.cn.
authors.forename: Runtao
authors.initials: R
authors.lastname: Li