title: Synthesis of 1-Amino-1H-Indenes via a Sequential Suzuki-Miyaura Coupling/Petasis Condensation Sequence.
abstract: An efficient and straightforward synthesis of 1-amino-1H-indenes is reported from 1,2-bis(boronates) via a sequential Suzuki-Miyaura coupling/Petasis cyclization reaction. Starting from the same monoboronic ester intermediates, an intermolecular version of this approach also afforded (Z)-α,β-unsaturated amino esters in moderate to good yields.
authors.affiliation: Organic and Biomolecular Chemistry Division, CSIR-Indian Institute of Chemical Technology , Tarnaka, Hyderabad 500 006, India.
authors.forename: Vankudoth
authors.initials: V
authors.lastname: Jayaram
authors.affiliation: Organic and Biomolecular Chemistry Division, CSIR-Indian Institute of Chemical Technology , Tarnaka, Hyderabad 500 006, India.
authors.forename: Tailor
authors.initials: T
authors.lastname: Sridhar
authors.affiliation: Organic and Biomolecular Chemistry Division, CSIR-Indian Institute of Chemical Technology , Tarnaka, Hyderabad 500 006, India.
authors.forename: Gangavaram V M
authors.identifier: 0000-0001-5638-788X
authors.initials: GV
authors.lastname: Sharma
authors.affiliation: Institut des Sciences Chimiques de Rennes, UMR 6226, CNRS-Université de Rennes 1 , 263, Avenue du Général Leclerc, Campus de Beaulieu, 35042 Rennes Cedex, France.
authors.forename: Fabienne
authors.initials: F
authors.lastname: Berrée
authors.affiliation: Institut des Sciences Chimiques de Rennes, UMR 6226, CNRS-Université de Rennes 1 , 263, Avenue du Général Leclerc, Campus de Beaulieu, 35042 Rennes Cedex, France.
authors.forename: Bertrand
authors.identifier: 0000-0003-0529-715X
authors.initials: B
authors.lastname: Carboni