title: Design of fluorogenic probes and fluorescent-tagged inhibitors for γ-glutamyl cyclotransferase.
authors.affiliation: Peptide Institute, Inc., Ibaraki, Osaka, 567-0085, Japan.
authors.forename: Taku
authors.identifier: http://orcid.org/0000-0002-7276-5614
authors.initials: T
authors.lastname: Yoshiya
authors.affiliation: Department of Clinical Oncology, Kyoto Pharmaceutical University, Kyoto, Kyoto, 607-8412, Japan.
authors.forename: Hiromi
authors.initials: H
authors.lastname: Ii
authors.affiliation: Peptide Institute, Inc., Ibaraki, Osaka, 567-0085, Japan.
authors.forename: Shugo
authors.initials: S
authors.lastname: Tsuda
authors.affiliation: Peptide Institute, Inc., Ibaraki, Osaka, 567-0085, Japan.
authors.forename: Masayoshi
authors.initials: M
authors.lastname: Mochizuki
authors.affiliation: Department of Urology, Shiga University of Medical Science, Otsu, Shiga, 520-2192, Japan.
authors.forename: Susumu
authors.initials: S
authors.lastname: Kageyama
authors.affiliation: Department of Clinical Oncology, Kyoto Pharmaceutical University, Kyoto, Kyoto, 607-8412, Japan.
authors.forename: Tatsuhiro
authors.initials: T
authors.lastname: Yoshiki
mesh_terms: D000818:Animals; D015195:Drug Design; D004791:Enzyme Inhibitors / Q000138:chemical synthesis / Q000737:chemistry / Q000494:pharmacology*; D005453:Fluorescence; D005456:Fluorescent Dyes / Q000138:chemical synthesis / Q000737:chemistry / Q000494:pharmacology*; D051379:Mice; D015394:Molecular Structure; D041681:NIH 3T3 Cells; D005722:gamma-Glutamylcyclotransferase / Q000037:antagonists & inhibitors* / Q000378:metabolism
chemical_list: D004791:Enzyme Inhibitors; D005456:Fluorescent Dyes; D005722:gamma-Glutamylcyclotransferase
keywords: GGCT; activity-based probe; cancer; fluorescence; inhibitor